Estazolam Tablet 1mg, 2mg Suppliers & Bulk Manufacturers

Available Forms: Tablets

Available Strengths: 1mg, 2mg

Reference Brands: Esilgan (EU), Eurodin (EU)

Category: Neurology

Estazolam is a benzodiazepine-class sedative-hypnotic primarily used for the short-term treatment of insomnia. It works by enhancing GABA activity in the central nervous system, producing calming and sleep-inducing effects.

Product Description:

Estazolam is a triazolobenzodiazepine hypnotic with an intermediate half-life of about ten to twenty-four hours. It enhances GABA-A receptor function like other benzodiazepines, and its hypnotic profile covers both sleep onset and maintenance. That profile suits patients who wake through the night, at the cost of more next-morning drowsiness than short-acting agents.

It is indicated for short-term treatment of insomnia, typically seven to ten days and rarely beyond a few weeks. Tolerance to its hypnotic effect develops with nightly use, dependence follows prolonged use, and stopping after regular use produces rebound insomnia, so tapering is advised. It is contraindicated in pregnancy. Additive respiratory and central nervous system depression with opioids and alcohol is the serious interaction, and CYP3A4 inhibitors raise exposure. Complex sleep behaviours such as sleep-driving have been reported.

Sourcing notes. Estazolam is a Schedule IV psychotropic under the 1971 UN Convention and Schedule IV in the US. International shipment requires import and export authorisations, with quota and reporting obligations. Registration is scattered — the US, Japan, China and parts of Europe and Latin America — and has been withdrawn in several markets where Z-drugs and newer hypnotics replaced it. Confirm registration and the controlled-substance pathway before quoting.